TC 2559 difumarate | CAS 212332-35-9

Element: difumarate 2559

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C-S » Chemicals » difumarate-PX77837

Identification

TC 2559 difumarate

CAS:

212332-35-9

EINECS:

Molecular Formula:

C₁₂H₁₈N₂O. 2C₄H₄O₄

MDL:

SMILES:

CCOC1=CN=CC(=C1)/C=C/CCNC.C(=C/C(=O)O)C(=O)O.C(=C/C(=O)O)C(=O)O

Synonym:

tc 2559 difumarate ; 4-(5-ethoxy-3-pyridinyl)-n-methyl-(3e)-3-buten-1-amine difumarate

Description

TC 2559 difumarate is a subtype-selective partial agonist for AChR α4β2 (EC₅₀ values are 0.18, 12.5, 14.0, > 30, > 100 and > 100 μM for α4β2, α4β4, α2β4, α3β4, α3β2 and α7 receptor subtypes, respectively). It displays selectivity for (α4)2(β2)3 receptor stoichiometry and enhanced CNS-PNS slectivity ratio.