SR 95531 Hydrobromide | CAS 104104-50-9

Element: hydrobromide 95531

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Identification

SR 95531 Hydrobromide

CAS:

104104-50-9

EINECS:

Molecular Formula:

C₁₅H₁₇ N₃ O₃ . Br H

MDL:

MFCD00055135

SMILES:

COC1=CC=C(C=C1)C2=NN(C(=N)C=C2)CCCC(=O)O.Br

Synonym:

1(6H)-Pyridazinebutanoicacid, 6-imino-3-(4-methoxyphenyl)-, monohydrobromide (9CI) ; Gabazine ; SR 95531 ; 1(6H)-Pyridazinebutanoicacid, 6-imino-3-(4-methoxyphenyl)-, hydrobromide (1:1)

Description

SR 95531 Hydrobromide is a selective GABA_A receptor antagonist. This compound displaces [3H]-GABA with a K_i of 150 nM. SR 95531 Hydrobromide selectively antagonizes GABA-induced Cl^- currents with little action on pentobarbitone-induced currents. SR 95531 Hydrobromide acts as a low affinity GlyR(glycine receptor)antagonist.