Chemical-Suppliers Chemical-Suppliers

N-Desmethyl Pirenzepine

×
Formula: C18H19N5O2
CAS: 63257-31-8
search Element: pirenzepine desmethyl
Page Content Identification Properties Suppliers Prices & Availability Get Quick Quote ☰

Identification

Structural Formula
N-Desmethyl Pirenzepine
CAS:
63257-31-8
EINECS:
Molecular Formula:
C18H19N5O2
MDL:
SMILES:
O=C(CN1CCNCC1)N1C2=CC=CC=C2C(=O)NC2=C1N=CC=C2
Synonym:
ls 822 ; n-desmethyl pirenzepine ; 5,11-dihydro-11-(1-piperazinylacetyl)-6h-pyrido[2,3-b][1,4]benzodiazepin-6-one ; 6h-pyrido(2,3-b)(1,4)benzodiazepin-6-one, 5,11-dihydro-11-(1-piperazinylacetyl)- ; 5,11-dihydro-11-(1-piperazinylacetyl)-6h-pyrido[2,3-β][1,4]benzodiazepin-6-one


Description

N-Desmethyl Pirenzepine is a metabolite of Pirenzepine. Pirenzepine is a selective antagonist for the M1 muscarinic receptor (mAChR) and is reported to block presynaptic M1 receptors as well as some reported inverse agonist activity. A study investigating the pharmacological characterization of the muscarinic receptors associated with ACh-induced pulmonary vasodilation in a rabbit model of pulmonary hypertension determined the IC50 to be 2.51x10-7M. Addtional research studies have investigated the role of Pirenzepine in the pathophysiology of myopia. Other M1 receptor antagonists offered include Telenzepine.


Suppliers

Santa Cruz Biotechnology, Inc.
212191
Get Quick Quote

Prices & Availability




Data is processed


x

Properties for N-Desmethyl Pirenzepine

Molecular Weight:
337.37576 g·mol−1
Density:
1.38 g/cm3
Boiling point:
496.7°C at 760 mmHg
Flash point:
254.2°C
x

Safety & Transport Information

coming up soon
x

Alternative Distributors of [N-Desmethyl Pirenzepine]

Producers or manufacturers change the product range from time to time. The following companies
have appeared as suppliers in the past / currently not verified

Clearsynth Canada INC.

x

Downloads

Mol File:
-/-
MSDS:
-/-




View related products













▲
▲