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Apstatin

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Formula: C23H33N5O5
CAS: 160470-73-5
search Element: apstatin
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Identification

Structural Formula
Apstatin
CAS:
160470-73-5
EINECS:
Molecular Formula:
C23H33N5O5
MDL:
MFCD01310909
SMILES:
CC(C(=O)N)NC(=O)C1CCCN1C(=O)C2CCCN2C(=O)C(C(CC3=CC=CC=C3)N)O
Synonym:
apstatin trifluoroacetate salt ; n-[(2s,3r)-3-amino-2-hydroxy-4-phenylbutanoyl]-l-prolyl-l-prolyl-l-alaninamide ; n-((2s,3r)-3-amino-2-hydroxy-4-phenylbutanoyl)-pro-pro-ala-nh2 ; apstatin hydrochloride ; n-(2s,3r)-ahpba-pro-pro-ala-nh2


Description

Apstatin is a selective inhibitor of aminopeptidase P (APP), with a Ki of 2.6 μM in rat lung membrane-bound APP. Apstatin is shown to increase Bradykinin-promoted cardioprotection in rats with artificially introduced myocardial infarctions by inhibiting the Bradykinin degradation action of APP. When combined with the angiotensin-converting enzyme inhibitors enalapril, lisinopril, or ramipril (sc-205833), decrease of myocardial infarction size was enhanced.


Suppliers

Santa Cruz Biotechnology, Inc.
201309
Dayang Chem (Hangzhou) Co.,Ltd.
DC248992
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Prices & Availability




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Properties for Apstatin

Molecular Weight:
459.54 g·mol−1
Density:
1.32 g/cm3
Melting point:
327.91° C
Boiling point:
864.33° C at 760 mmHg
Solubility:
Soluble in water (>25 mg/ml), and DMSO (20 mg/ml).
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Safety & Transport Information

Storage temperature :
-20°C
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Alternative Distributors of [Apstatin]

Producers or manufacturers change the product range from time to time. Currently there are no other manufacturers known.
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Downloads

Mol File:
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MSDS:
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